Pertuzumab biosimilars

Anti-HER2 antibody used with trastuzumab in HER2-positive breast cancer, with the first biosimilar approved in the US in November 2025 and three Indian manufacturers permitted since 2024.

Reference product Perjeta (Roche) · Monoclonal antibody · Target HER2 (domain II) · ATC L01FD02 · Oncology
FDAproducts approved, 1 interchangeable1
EMAproducts authorised1
CDSCOpermissions3
EDEregistered in the UAE0

About pertuzumab

Molecule

Humanised IgG1 kappa monoclonal antibody of about 148 kDa, produced in Chinese hamster ovary cells, directed against extracellular domain II of HER2, a different site from the domain IV epitope bound by trastuzumab.

Mechanism of action

Blocks HER2 from forming ligand-dependent dimers with other HER family receptors, particularly HER3, which trastuzumab does not prevent; the two antibodies together give a more complete blockade of HER2 signalling. It also mediates antibody-dependent cellular cytotoxicity.

Pharmacokinetics

Intravenous infusion; half-life about 18 days, linear pharmacokinetics at clinical doses, steady state after the first maintenance dose. A subcutaneous fixed combination with trastuzumab and hyaluronidase exists for the reference product.

Dosing and presentations

840 mg loading dose then 420 mg every three weeks with trastuzumab and chemotherapy, as 420 mg/14 mL (30 mg/mL) concentrate for infusion in single-dose vials.

Approved indications
  • HER2-positive metastatic breast cancer with trastuzumab and docetaxel
  • Neoadjuvant treatment of HER2-positive early breast cancer at high risk of recurrence
  • Adjuvant treatment of HER2-positive early breast cancer at high risk of recurrence
Immunogenicity

Anti-pertuzumab antibodies are rare and not clinically relevant. Comparative programmes use analytical similarity with attention to HER2 domain II binding and ADCC, a pharmacokinetic study, and a comparative efficacy study in the neoadjuvant setting with pathological complete response as the endpoint, in combination with trastuzumab and chemotherapy.

Reference product: Perjeta

Perjeta was licensed by FDA on 8 June 2012 (BLA 125409) and authorised in the EU on 4 March 2013 (EMEA/H/C/002547). The first Indian biosimilar was permitted to Zydus in April 2024, and Henlius's Poherdy became the first US biosimilar in November 2025, interchangeable on licensure, followed by EU authorisation through Organon in April 2026. Roche's subcutaneous fixed combination with trastuzumab, Phesgo, has no biosimilar.

Sources: Purple Book (S016), EMA medicines data (S017), CDSCO lists (S011, S012, S013).

Why pertuzumab matters for biosimilar developers

Pertuzumab is the natural second step for any developer with a trastuzumab biosimilar, since the two are given together and the neoadjuvant study design is the same. India moved first: Zydus in 2024, Intas and Enzene in 2025, all at the 420 mg/14 mL presentation, while the West has a single product from Henlius. Roche's defence is Phesgo, the subcutaneous combination, which has no biosimilar in any market.

Sources: Perjeta summary of product characteristics (EMA) and US prescribing information (FDA).

Approvals by year

20132014201520162017201820192020202120222023202420252026FDAPoherdy (2025)EMAPoherdy (2026)CDSCOZydus Lifesciences (INN only) (2024)Intas Pharmaceuticals (INN only), Enzene Biosciences (INN only) (2025)Intas Pharmaceuticals (INN only), Enzene Biosciences (INN only) (2025)EDE
FDANov 2025Poherdy
EMAApr 2026Poherdy
CDSCOApr 2024Zydus Lifesciences (INN only)
EDEnonenot listed

Regulatory register

RegulatorBrandHolder or applicantApprovedApplication or permissionUS licenceStatusSource
FDAPoherdyShanghai Henlius Biotech, Inc.Nov 2025761450InterchangeableApprovedS001, S016
EMAPoherdyOrganon N.V.Apr 2026EMEA/H/C/006583ApprovedS017
CDSCOZydus Lifesciences (INN only)Zydus Lifesciences LimitedApr 2024MF/BIO/24/000041ApprovedS011
CDSCOIntas Pharmaceuticals (INN only)Intas Pharmaceuticals LtdJan 2025MF/BIO/25/000006ApprovedS011
CDSCOEnzene Biosciences (INN only)Enzene Biosciences LtdJun 2025MF/BIO/25/000085ApprovedS011

CDSCO lists permissions by firm and INN, not brand. The UAE directory does not publish registration numbers.

Regulatory pathway by market

Requirements for a pertuzumab biosimilar under the guidance in force in September 2026.

FDA, United StatesEMA, European UnionCDSCO, IndiaEDE, UAE
Legal pathwaySection 351(k) of the Public Health Service Act (BPCIA 2009)Article 10(4) of Directive 2001/83/EC; centralised procedure is mandatory for biotechnology productsGuidelines on Similar Biologics (CDSCO and DBT, 2016, in force); revised draft published May 2025Registration through the Emirates Drug Establishment; the public directory does not distinguish biosimilars from other biologicals
Reference productUS-licensed reference; a non-US comparator may be used with analytical and PK bridgingEU-authorised reference; a non-EEA comparator may be used with bridging dataProduct licensed in India, or if not, one licensed in an ICH country, with justificationNot stated in the public directory; registration relies on assessment by reference regulators
Comparative clinical studyDraft guidance (October 2025): comparative analytical assessment plus a PK similarity study and immunogenicity assessment; a comparative efficacy study is generally not neededReflection paper adopted March 2026: a comparative efficacy trial can be waived when analytical and PK comparability is sufficientComparative PK/PD study and a comparative safety and efficacy study are generally expected, followed by a post-marketing studyAssessed on the dossier accepted by the reference regulator
InterchangeabilityA separate designation permitting pharmacy-level substitution; switching studies generally not required under the June 2024 draftEMA and HMA statement (September 2022): EU biosimilars are interchangeable with their reference; substitution rules are set by each member stateNot defined in the guidelinesNot defined
NamingINN plus a four-letter suffixINN, identical to the reference; brand name and batch recorded for pharmacovigilanceINN with the brand nameBrand name as registered

Sources: FDA draft guidance on comparative efficacy studies (October 2025) and interchangeability (June 2024); EMA reflection paper EMA/CHMP/BMWP/60916/2025 (March 2026) and EMA/HMA statement on interchangeability (September 2022); CDSCO Guidelines on Similar Biologics 2016 and 2025 draft (S009, S010); EDE directory (S018).

EvySaif prepares the comparative evidence plan and the regional dossier strategy for pertuzumab programmes. Regulatory strategy consulting

Presentations and concentration

A single presentation, 420 mg in 14 mL (30 mg/mL) concentrate for infusion. The subcutaneous combination with trastuzumab (Phesgo) exists only for the reference product.

ProductFDAEMACDSCOEDE
Poherdy HLX11
420 mg/14 mL vial
see SmPC··
Zydus pertuzumab··
420 mg/14 mL (30 mg/mL) vial
·
Intas pertuzumab··
420 mg/14 mL (30 mg/mL) vial
·
Enzene Biosciences pertuzumab··
420 mg/14 mL (30 mg/mL) vial
·

Sources: Purple Book (S016), CDSCO permission lists (S011 to S014), EDE directory (S018). EU presentations are listed in each product's SmPC.

Developers by market

DeveloperProductFDAEMACDSCOEDE
Shanghai Henlius BiotechPoherdy··
Zydus LifesciencesZydus pertuzumab···
Intas PharmaceuticalsIntas pertuzumab···
Enzene Biosciences (Alkem)Enzene Biosciences pertuzumab···

Entering a market where a competitor is already listed changes the evidence and pricing conversation. EvySaif's global value dossier and HTA submission work covers that side.

Products

Questions

How many pertuzumab biosimilars has FDA approved?

One: Poherdy from Shanghai Henlius, approved on 13 November 2025 and designated interchangeable on the same day.

Which pertuzumab biosimilars are authorised in the European Union?

One: Poherdy, authorised on 23 April 2026 with Organon as the holder.

Is there a pertuzumab biosimilar approved in India?

Yes, three. CDSCO permitted Zydus Lifesciences in April 2024 (with early breast cancer added in August 2024), Intas Pharmaceuticals in January 2025 (neoadjuvant indication added February 2026) and Enzene Biosciences in June 2025.

Which pertuzumab biosimilars are registered in the UAE?

None yet in the Emirates Drug Establishment directory; Perjeta and Phesgo are registered.

Is there a biosimilar of Phesgo?

No. The subcutaneous fixed combination of pertuzumab, trastuzumab and hyaluronidase is a separate product with its own patents and no biosimilar in any market.

Which comparative efficacy study do regulators accept for pertuzumab?

A neoadjuvant study in HER2-positive early breast cancer, in combination with trastuzumab and chemotherapy, with total pathological complete response as the primary endpoint, supported by pharmacokinetic equivalence and analytical comparability of domain II binding and ADCC.

Work with EvySaif on pertuzumab

Pertuzumab biosimilar landscape report

The register on this page as a delivered document: every approval, holder, presentation and pathway requirement across FDA, EMA, CDSCO and the Gulf, updated to the month, with the sources attached.

Request the landscape report

Regulatory gap assessment

For a developer deciding whether and where to file: a review of your analytical, PK and clinical package against what each regulator expects for pertuzumab, with the gaps ranked and a filing sequence recommended.

About the gap assessment

Sources

Planning pertuzumab biosimilar development?

EvySaif can help assess your regulatory pathway, clinical evidence requirements and market-entry strategy across India, UAE and other target markets.

Talk to a biosimilar regulatory consultant
Data current to September 2026.